Tesofensine | CAS No. 195875-84-4

Tesofensine

Basic Information

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CAS Number

195875-84-4

Molecular Formula

C17H23Cl2NO

Molecular Weight

328.28 g/mol

Chemical Classification

Basic Chemical Raw Materials Organic Chemicals Ethers

Basic Chemical Raw Materials Organic Chemicals Heterocyclic Compounds

Pharmaceutical Chemicals Pharmaceutical Intermediates Heterocyclic Intermediates

Agricultural Chemicals Pesticides Herbicides

Basic Physical Properties

SMILES

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CCOC[C@H]1[C@H]2CC[C@H](N2C)C[C@@H]1c1ccc(c(c1)Cl)Cl

InChI

InChI=1S/C17H23Cl2NO/c1-3-21-10-14-13(9-12-5-7-17(14)20(12)2)11-4-6-15(18)16(19)8-11/h4,6,8,12-14,17H,3,5,7,9-10H2,1-2H3/t12-,13+,14+,17+/m0/s1

InChIKey

VCVWXKKWDOJNIT-ZOMKSWQUSA-N

LogP

4.596200000000005

Topological Polar Surface Area

12.47 Å²

Hydrogen Bond Donor/Acceptor

0 / 2

Synonyms & References

English

Tesofensine
(1R,2R,3S,5S)-3-(3,4-Dichlorophenyl)-2-(ethoxymethyl)-8-methyl-8- azabicyclo[3.2.1]octane
NS 2330
(1S,3S,4R,5R)-3-(3,4-dichlorophenyl)-4-(ethoxymethyl)-8-methyl-8-azabicyclo[3.2.1]octane
(1R,2R,3S,5S)-3-(3,4-dichlorophenyl)-2-(ethoxymethyl)-8-methyl-8-azabicyclo[3.2.1]octane

MDL Number

MFCD18633271

FAQ

What is Tesofensine (CAS: 195875-84-4)?

Tesofensine (CAS: 195875-84-4) is a pharmacological compound that acts as a dual-norepinephrine and serotonin uptake inhibitor with weak anticholinergic activity. It is primarily used in the treatment of depression and attention deficit hyperactivity disorder (ADHD).

What are the main uses of Tesofensine (CAS: 195875-84-4)?

Tesofensine (CAS: 195875-84-4) is mainly used as an antidepressant and for the treatment of attention deficit hyperactivity disorder (ADHD). It is also being studied for potential uses in other neurological disorders.

Is Tesofensine (CAS: 195875-84-4) safe?

Tesofensine (CAS: 195875-84-4) is generally considered safe when used as directed. However, it may cause side effects such as dry mouth, constipation, and urinary retention. It is important to follow the prescribed dosage and consult a healthcare provider regarding any concerns.

How should Tesofensine (CAS: 195875-84-4) be stored?

Tesofensine (CAS: 195875-84-4) should be stored in a tightly closed container at room temperature, protected from light and moisture. It should be kept out of reach of children and pets.