tert-Butyl 4-chloro-5-methoxypyridin-3-ylcarbamate
CAS Number:
1045858-17-0
Molecular Formula:
C11H15ClN2O3
One-pot two-step radioiodination based on copper-mediated iododeboronation and azide–alkyne cycloaddition reaction
Literature Information
Publication Date
2023-12-18
DOI
10.1039/D3CC04787C
Impact Factor
6.222
Authors
Yuto Kondo, Ryota Chisaka, Yasunao Hattori, Hidekazu Kawashima, Hiroyuki Yasui
View Original
Abstract
This methodology demonstrates the ability to sequentially regulate copper-mediated radioiododeboronation and an azide–alkyne cycloaddition reaction, which facilitates the continuous incorporation of reagents into the reaction system and mediates the integration of the purification steps into the final process. Additionally, this reaction is suited to be conducted under mild conditions and yields target compounds through potent radiochemical conversions.
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Source Journal
Chemical Communications
CiteScore:
8.6
Self-citation Rate:
4.7%
Articles per Year:
2458
ChemComm publishes urgent research which is of outstanding significance and interest to experts in the field, while also appealing to the journal’s broad chemistry readership. Our communication format is ideally suited to short, urgent studies that are of such importance that they require accelerated publication. Our scope covers all topics in chemistry, and research at the interface of chemistry and other disciplines (such as materials science, nanoscience, physics, engineering and biology) where there is a significant novelty in the chemistry aspects. Major topic areas covered include: Analytical Chemistry Catalysis Chemical Biology and medicinal chemistry Computational Chemistry and Machine Learning Energy and sustainable chemistry Environmental Chemistry Green Chemistry Inorganic Chemistry Materials Chemistry Nanoscience Organic Chemistry Physical Chemistry Polymer Chemistry Supramolecular Chemistry
Recommended Compounds
5-(2-Methyl-1,3-thiazol-4-yl)-2-thiophenesulfonyl chloride
CAS Number:
215434-25-6
Molecular Formula:
C8H6ClNO2S3
-1,2-cyclohexanediamine structure](https://static.chemtradehub.com/structs/928/928769-12-4-a4f0.webp "N,N'-Bis[3-(2-methoxyphenyl)-2-hydroxybenzyl](1R,2R)-1,2-cyclohexanediamine structure")
N,N'-Bis[3-(2-methoxyphenyl)-2-hydroxybenzyl](1R,2R)-1,2-cyclohexanediamine
CAS Number:
928769-12-4
Molecular Formula:
C34H38N2O4
![1-(2-Chlorophenyl)-6-[(2S)-3,3,3-trifluoro-2-methylpropyl]-1,7-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one structure](https://static.chemtradehub.com/structs/794/794568-91-5-0c34.webp "1-(2-Chlorophenyl)-6-[(2S)-3,3,3-trifluoro-2-methylpropyl]-1,7-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one structure")
1-(2-Chlorophenyl)-6-[(2S)-3,3,3-trifluoro-2-methylpropyl]-1,7-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one
CAS Number:
794568-91-5
Molecular Formula:
C15H12ClF3N4O
8-Methyl-2-pyridin-4-ylquinoline-4-carboxylic acid
CAS Number:
107027-42-9
Molecular Formula:
C16H12N2O2
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