Tiagabine(CAS: 115103-54-3)

Tiagabine is a selective GABA transaminase inhibitor, used as an anticonvulsant in the treatment of epilepsy. It has a chemical formula of C14H18N2O2. Tiagabine is known for its ability to increase GABA levels in the brain, which is crucial for inhibiting neuronal excitability and preventing seizures.

Tiagabine is primarily used as an anticonvulsant to treat partial seizures in epileptic patients. It can be administered orally and is often used in combination with other anticonvulsant drugs to better control seizures.

Tiagabine can be considered safe when used under medical supervision. However, it requires close monitoring due to potential side effects such as dizziness, headache, and emotional changes. Patients should avoid operating heavy machinery and driving until they are aware of their response to the medication. Protective measures include wearing gloves and eye protection during handling.

Tiagabine should be stored in a tightly closed container at room temperature (15-30°C) and away from direct sunlight. It should be kept in a cool, dry place to prevent degradation. Avoid storing it in high humidity or near heat sources. The container should be child-proof to prevent accidental ingestion.